Bivalent Ligands for the Serotonin 5-HT3 Receptor
نویسندگان
چکیده
منابع مشابه
High-affinity fluorescent ligands for the 5-HT3 receptor
The synthesis, photophysical and biological characterization of a small library of fluorescent 5-HT(3) receptor ligands is described. Several of these novel granisetron conjugates have high quantum yields and show high affinity for the human 5-HT(3)AR.
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ژورنال
عنوان ژورنال: ACS Medicinal Chemistry Letters
سال: 2011
ISSN: 1948-5875,1948-5875
DOI: 10.1021/ml2000388